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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T67755 | Protein kinase G inhibitor-1 | PKA | |
Protein kinase G inhibitor-1 is a potent Protein kinase G inhibitor, IC50= 0.9 uM. | |||
T9940 | Protein kinase G inhibitor-2 | Others | |
Protein kinase G inhibitor-2 exhibits antibacterial, antiviral, and antitumor activities. | |||
TP1902L1 | G-Protein antagonist peptide acetate | Adrenergic Receptor | |
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide acetate inhibits the activation of Gi or Go by M2 muscarinic cho... | |||
TP1902 | G-Protein antagonist peptide | ||
Substance P-related peptide that inhibits binding of G proteins to their receptors. Competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors. | |||
T14898 | CCG-63808 | GTPase | |
CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins. CCG-63808 dose-dependently inhibits the TR-FRET signal between RGS4-AF488 and Tb-Gαo with IC50 values of 1.9 μM. | |||
T14897 | CCG-63802 | GTPase | |
CCG-63802 is a reversible inhibitor of the regulator of G-protein signaling (RGS) protein and has the greatest potency at RGS4. | |||
TP2254 | GTP-Binding Protein Fragment, G alpha | Others | |
Using specific antisera raised against synthetic peptides, we find that three distinct GTP-binding protein alpha subunits remain bound to the plasma membrane even after activation with nonhydrolyzable GTP analog. Trypsin... | |||
T8818 | TC-G 1005 | GPCR19 | |
TC-G 1005 is a potent and selective GPBA agonist (EC50 :0.72 nM; hTGR5). Selective for TGR5 over FXR (farnesoid X receptor). Increases plasma GLP-1 levels and reduces blood glucose in mice. Orally available. | |||
T7428 | SBI-115 | GPCR19 | |
SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5 | |||
T4083 | BAR501 | BAR 501 | GPCR19 |
BAR501 is an effective and specific GPBAR1 agonist (EC50: 1 μM). | |||
TQ0252 | BAR502 | FXR , GPCR19 , Autophagy | |
BAR502 is a dual GPBAR1 and FXR agonist (IC50s: 0.4 μM and 2 μM). | |||
T20731 | Brilliant blue G-250 | BBG,Acid blue 90, Coomassie Brilliant Blue G,Brilliant Blue G | P2X Receptor |
Brilliant blue G-250 (Acid blue 90, Coomassie Brilliant Blue G) is an antagonist of the P2X7 purinergic receptor. | |||
T4352 | SB756050 | SB-756050,SB 756050 | GPCR19 |
SB756050 is a specific TGR5 agonist. | |||
T2088 | APD668 | APD 668 | GPR , P450 , Potassium Channel |
APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119, respectively. | |||
T6434 | CCG-50014 | CCG 50014 | GTPase |
CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM. | |||
T16378 | Ogerin | Others , 5-HT Receptor , Adenosine Receptor | |
Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice. Ogerin displays inverse agonist and antagonist activity (Ki, 220 nM) at A2A receptor and weak an... | |||
T1793 | MBX-2982 | GPR | |
MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes. | |||
T21874 | CID 2745687 | GPR | |
CID 2745687 is a GPR35 antagonist that inhibited the effects at human GPR35 of cromolyn disodium and zaprinast, two agonists that share an overlapping binding site. | |||
T6843 | GDC-0623 | G-868,GDC0623,RG 7421,MEK inhibitor 1 | Apoptosis , MEK |
GDC-0623 (RG 7421) is a potent and ATP-uncompetitive MEK1 inhibitor with Ki of 0.13 nM. Phase 1. | |||
T1824 | TGR5 Receptor Agonist | GPCR19 | |
TGR5 is a potent TGR5(GPCR19) agonist. | |||
T2701 | GSK1292263 | GPR | |
GSK1292263 is a GPR119 agonist and has been investigated for the treatment of DIABETES MELLITUS, TYPE 2. | |||
T22996 | ML-191 | ERK | |
ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2. | |||
T6313 | Go 6983 | Goe 6983 | PKC |
Go 6983 is a pan-PKC inhibitor targeting PKCα, PKCβ, PKCγ, PKCδ, and PKCζ, exhibiting IC50 values of 7 nM, 7 nM, 6 nM, 10 nM, and 60 nM, respectively. | |||
T4626 | TC-O 9311 free base | GPR | |
TC-O 9311 is a potent GPR139 agonist. | |||
T22408 | Proflavine | 3,6-Diaminoacridine | Antibacterial |
Proflavine (3,6-Diaminoacridine) (3,6-Diaminoacridine) is a disinfectant bacteriostatic against many gram-positive bacteria and is a topical antiseptic used mainly in wound dressings. | |||
T7156 | NIBR189 | EBI2/GPR183 | |
NIBR189 is a potent and selective antagonist of EBI2 (GPR183) receptor (IC50 of 11 and 15 nM for human and mouse EBI2 receptors, respectively) | |||
T8329 | AR 231453 | GPR | |
AR 231453 is a selective and orally available GPR119 agonist,can stimulate β-cell replication and improve islet graft function. | |||
T2036 | 6-OAU | GTPL5846 | GPR |
6-OAU (GTPL5846)(GTPL5846; 6-n-octylaminouracil) is a surrogate agonist of GPR84; activates human GPR84 in the presence of Gqi5 chimera in HEK293 cells with an EC50 of 105 nM in the PI assay. | |||
T8975 | PSB-SB-487 | Cannabinoid Receptor | |
PSB-SB-487 is antagonist of GPR55. | |||
T8571 | ML-184 | CID2440433 | Cannabinoid Receptor |
ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM. | |||
T3119 | JNJ-63533054 | JNJ 63533054 | GPR |
JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM. | |||
T3176 | APD597 | JNJ-38431055 | GPR |
APD597 (JNJ-38431055) is a GPR119 agonist, used in the treatment of type 2 diabetes. | |||
T21623 | AS1269574 | AS 1269574 | GPR , TRP/TRPV Channel |
AS1269574 is a potent, orally available GPR119 agonist. AS1269574(AS 1269574) has the potential for the research of type 2 diabetes. | |||
T22103 | ML-193 | CID 1261822 | Cannabinoid Receptor |
ML-193 (CID 1261822) is a potent and selective GPR55 antagonist( IC50 : 221 nM). It shows more than 27-fold selectivity for GPR55 over GPR35, CB1 and CB2, and can improve the motor and the sensorimotor deficits of Parkin... | |||
T23204 | PSN 375963 | PSN 375963 hydrochloride | GPR |
PSN 375963 (PSN 375963 hydrochloride) hydrochloride is a synthetic agonist of the endogenous ligand for GPR119. | |||
T9317 | TAK-041 | NBI-1065846 | GPR |
TAK-041 (NBI-1065846) is a potent and selective GPR139 agonist. | |||
T0438 | Proflavine Hemisulfate | 3,6-Diaminoacridine hemisulfate,Proflavin hemisulfate | Others , Potassium Channel , DNA , Thrombin , Antibacterial , Autophagy |
Proflavine Hemisulfate (3,6-Diaminoacridine hemisulfate) is the hemisulfate salt form of proflavine, an acridine-derived fluorescent contrast and disinfectant agent that can potentially be used for cellular imaging and a... | |||
T4494 | CLOZAPINE N-OXIDE | Dopamine Receptor , 5-HT Receptor , AChR , Drug Metabolite | |
Clozapine N-oxide is the major metabolite of Clozapine and is blood-brain barrier permeable. Clozapine N-oxide is an agonist of DREADDs and activates the DREADD receptors hM3Dq and hM4Di. Clozapine N-oxide is also a dopa... | |||
T4478 | CID 16020046 | C390-0219 | Cannabinoid Receptor |
CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast. | |||
T12883 | Fezagepras | PBI-4050,Setogepram | GPR |
Fezagepras (Setogepram) is an orally active GPR40 agonist and is an antagonist or inverse agonist of GPR84 with anti-inflammatory, anti-fibrotic, and anti-proliferative actions. | |||
T28073 | MLS1547 | MLS000051547,MLS 1547,MLS-1547 | Dopamine Receptor |
MLS1547 (MLS000051547) is a highly efficacious agonist of G protein-biased dopamine D2 receptor with a Ki of 1.2 μM. MLS1547 stimulates D2R G protein-mediated signaling with EC50 of 0.37 μM in a calcium mobilization assa... | |||
T10363 | Arazine | N-Acetyl-S-farnesyl-L-cysteine | Others |
Arazine (N-Acetyl-S-farnesyl-L-cysteine) can be a a substrate for isoprenylcysteine methyltransferase by competing with prenylated G protein or its receptors site. Arazine is a cell-permeable modulator of G protein and G... | |||
T36036 | CAY10786 | GPR52 antagonist-1 | GPR |
CAY10786 (GPR52 antagonist-1) is an antagonist of G protein-coupled receptor 52 (GPR52, IC50 = 0.63 μM). | |||
T16519L | BIM-46187 4HCl | PH-064 4HCl | Others |
BIM-46187 4HCl (PH-064 4HCl) is a heterotrimeric G-protein complex inhibitor. | |||
T13807 | OSIP-486823 | CP248 | Microtubule Associated , PKA |
OSIP-486823(CP248) is a novel and potent microtubule disruptor with affinity for both protein kinase G (PKG) and microtubules. | |||
T7281 | F-15599 | 5-HT Receptor | |
F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM). | |||
T50088 | N-phenylthiophene-2-carboximidamide | Others | |
N-phenylthiophene-2-carboximidamide is a thiophene derivative that functions as an inhibitor of protein tyrosine kinases (PTKs) and a ligand for G protein-coupled receptors (GPCRs). | |||
T5100 | DJ-V-159 | DJ-V159 | GPR , Androgen Receptor |
DJ-V-159 is a GPRC6A agonist, targeting the G protein-coupled receptor family C group 6 member A (GPRC6A). | |||
T7312 | AX20017 | Others , Antibacterial | |
AX20017 is a small-molecule protein kinase G (PknG) inhibitor(IC50 : 0.39 μM). It acts by blocking the proliferation of M. tuberculosis. | |||
T5422 | CID 1375606 | CID-1375606,CID1375606 | Others |
CID 1375606 is a surrogate agonist of orphan G protein-coupled receptor GPR27. characterized by a high level of conservation among vertebrates and a predominant expression in the central nervous system. |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6512 | G-418 disulfate | Geneticin,G418 Sulfate,Antibiotic G-418 sulfate,Geneticin sulfate | Antibacterial , Antibiotic |
G-418 disulfate (Geneticin sulfate) is an aminoglycoside antibiotic, an inhibitor of protein synthesis with eukaryotic selectivity. G-418 disulfate blocks peptide synthesis by inhibiting peptide chain elongation. | |||
T5077 | Deoxycholic acid sodium salt | Sodium deoxycholate,Sodium Desoxycholate | Endogenous Metabolite , GPCR19 |
Deoxycholic acid sodium salt (Sodium deoxycholate) can activate the G protein-coupled bile acid receptor TGR5 that stimulates brown adipose tissue (BAT) thermogenic activity. | |||
T2965 | Deoxycholic acid | Cholorebic,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic | Endogenous Metabolite , GPCR19 |
Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate. It is usually conjugated with glycine or taurine. Deoxycholic acid acts as a detergent to solubilize fats for intestinal absorptio... | |||
TN2268 | Tetrahydromagnolol | Cannabinoid Receptor , GPR , GABA Receptor | |
Tetrahydromagnolol can activate cannabinoid (CB) receptors. | |||
T0700 | Ursodeoxycholic acid | UDCA,Ursodiol | Potassium Channel , Endogenous Metabolite |
Ursodeoxycholic acid (UDCA) can be used to dissolve gallstones and reduce cholesterol absorption. | |||
T2968 | Hyodeoxycholic acid | NSC 60672,α-Hyodeoxycholic Acid,HDCA | FXR , Endogenous Metabolite , GPCR19 |
Hyodeoxycholic acid (NSC 60672) has been used in trials studying the treatment of Hypercholesterolemia. | |||
T29078 | Ursodeoxycholic acid sodium | UDCA Na,UDCA sodium,Sodium Ursodeoxycholate,Ursodiol sodium,Ursodeoxycholic Acid (sodium salt),Ursodeoxycholate sodium | FXR , Endogenous Metabolite , GPCR19 |
Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities. Ursodeoxycholic acid sodium acts as signaling molecule, exerting it... | |||
T14046 | Anandamide | (5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide | Cannabinoid Receptor , Endogenous Metabolite |
Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but also other targets (e.g., GPR18/GPR55) in the central nervous sy... | |||
T0508 | γ-Aminobutyric acid | Gamma-aminobutyric acid,4-Aminobutyric acid,GABA,4-Aminobutanoic acid,Piperidic acid | GABA Receptor , Endogenous Metabolite |
γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system. | |||
T4839 | Ac-Ala-OH | N-Acetylalanine,N-Acetyl-L-alanine | Others , Endogenous Metabolite |
Ac-Ala-OH (N-Acetyl-L-alanine) is a substrate for Guanine nucleotide-binding protein G(I)/G(S)/G(O) gamma-2 subunit, Myelin basic protein, GTP-binding nuclear protein Ran, Tropomyosin alpha 4 chain, HIV-1 Rev binding pro... | |||
T20003 | Acridone | Antibacterial , ABC | |
Acridone could induce cell apoptosis, inhibited ABCG2 (ATP-binding cassette sub-family G member 2) protein, and adjusted hormone level. | |||
T3S1612 | Kuwanon G | Moracenin B,Kuwanone G | Phosphatase , Antibacterial , Bombesin Receptor , AChR , AChE , Glucosidase |
1. Kuwanon G (Moracenin B) as dual inhibitors of PTP1B and α-glucosidase enzymes, as well as insulin sensitizers, it may potentially be utilized as an effective treatment for Type II diabetes mellitus. 2. Kuwanon G has a... | |||
T3232 | Higenamine hydrochloride | Higenamine HCl,Demethylcoclaurine hydrochloride,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride | Adrenergic Receptor |
Higenamine hydrochloride (norcoclaurine HCl) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein–coupled receptors, and are the most prominent... | |||
T5065 | GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD | Monosodium-GMP,cGMP sodium salt,Cyclic GMP | PKA |
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD (cGMP sodium salt) , also known as cGMP, is a cellular regulatory agent and has been described as a second messenger. Its levels increase in response to a variety of hormones, inc... | |||
T3929 | Kaurenoic acid | Kauren-19-Oic Acid,kaurenoate,kaur-16-en-18-oic acid | Others |
Kaurenoic acid (kaurenoate) has anti-inflammatory potential in acetic acid-induced colitis, decreases in MDA level. Kaurenoic acid exerts a uterine relaxant effect acting principally through calcium blockade and in part,... | |||
T17273 | YM-254890 | Others | |
YM-254890 inhibits platelet aggregation induced by ADP by blocking the P2Y1 signal transduction pathway (IC50: below 0.6 μM). YM-254890 is a selective Gαq/11 protein inhibitor. YM-254890 displays no inhibition of other G... | |||
T73876 | Sanggenon G | ||
Sanggenon G, a cell-permeable and potent inhibitor of X-linked inhibitor of apoptosis protein (XIAP), specifically binds to the XIAP BIR3 domain with a binding affinity of 34.26 μM, thereby enhancing caspase activation [... | |||
TN5580 | Rediocide A | ||
Rediocide A, an insecticide, can inhibit calcium mobilization in Drosophila G-protein- coupled receptors (GPCR)s other than methuselah, it can induce GPCR desensitization and internalization, and such effects are mediate... | |||
T38331 | Commendamide | ||
Commendamide is a natural bacterial product that was discovered in a screen for commensal bacteria effector genes (Cbegs). Cbeg12 is a bacterial effector gene that encodes for its production. Commendamide is structurally... | |||
T21500 | Sphingosine-1-phosphate | S1P | Endogenous Metabolite , S1P Receptor , LPL Receptor |
Sphingosine-1-phosphate (S1P) is an agonist for S1P1-5 receptors and a ligand for GPR3, GPR6, GPR12.Sphingosine-1-phosphate is an intracellular second messenger that mobilises Ca2+ as an extracellular ligand for G-protei... | |||
T38069 | Aquastatin A | ||
Aquastatin A is a fungal metabolite originally isolated fromF. aquaeductuumthat has diverse biological activities.1It is active againstS. aureus(MIC = 32 μg/ml) and inhibits enoyl-acyl carrier protein reductase (Fabl; IC... |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-01885 | Human RSV (B1) glycoprotein G/RSV-G Protein (His) | RSV | HEK293 Cells |
Human RSV (B1) glycoprotein G/RSV-G Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27 kDa and the accession number is O36633-1. | |||
TMPY-01082 | Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (95% Homology) (His) | RSV | HEK293 Cells |
Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (95% Homology) (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.7 kDa and the accession num... | |||
TMPY-02283 | Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (93% Homology) (His) | RSV | Baculovirus Insect Cells |
Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (93% Homology) (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 26.3 kDa and the accession n... | |||
TMPY-00105 | Recombinant Protein G | E. coli | |
Protein G is a bacterial cell wall protein expressed at the cell surface of certain group C and group G Streptococcal strains. It has affinity for both Fab- and Fc-fragments of human IgG by independent and separate bindi... | |||
TMPY-06469 | Human respiratory syncytial virus (RSV) (B, strain 18537) glycoprotein G Protein (His) | RSV | HEK293 Cells |
Human respiratory syncytial virus (RSV) (B, strain 18537) glycoprotein G Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.40 kDa and the accession number is P20896. | |||
TMPY-06474 | Human respiratory syncytial virus (RSV) (strain A2) glycoprotein G Protein (His) | RSV | HEK293 Cells |
Human respiratory syncytial virus (RSV) (strain A2) glycoprotein G Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.97 kDa and the accession number is P03423. | |||
TMPY-05686 | Human respiratory syncytial virus (RSV) glycoprotein G Protein (aa 64-321, His) | RSV | HEK293 Cells |
Human respiratory syncytial virus (RSV) glycoprotein G Protein (aa 64-321, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 29.59 kDa and the accession number is A0A076FRQ0. | |||
TMPY-06111 | Human respiratory syncytial virus (RSV) (subtype A, strain Long) glycoprotein G Protein (His) | RSV | HEK293 Cells |
Human respiratory syncytial virus (RSV) (subtype A, strain Long) glycoprotein G Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27 kDa and the accession number is P208... | |||
TMPY-05636 | G-CSF Protein, Mouse, Recombinant | Mouse | HEK293 Cells |
G-CSF Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 19 kDa and the accession number is P09920. | |||
TMPY-04829 | G-CSF Protein, Human, Recombinant | Human | HEK293 Cells |
G-CSF Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 18.7 kDa and the accession number is P09919-2. | |||
TMPY-02312 | CSF3R/G-CSFR Protein, Human, Recombinant (His) | Human | HEK293 Cells |
CSF3R/G-CSFR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 68 kDa and the accession number is Q99062-1. | |||
TMPY-00300 | Hendra virus (HeV) (isolate Horse/Autralia/Hendra/1994) Glycoprotein Protein (hFc) | HEV | HEK293 Cells |
Hendra virus (HeV) (isolate Horse/Autralia/Hendra/1994) Glycoprotein Protein (hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 86.3 kDa and the accession number is O89343. | |||
TMPH-00510 | DT3C Protein, Recombinant (His) | Corynephage beta | E. coli |
DT3C Protein, Recombinant (His) is expressed in E. coli. | |||
TMPK-00876 | G-CSFR/CD114 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
The Granulocyte Colony-Stimulating Factor (G-CSF) receptor, a member of the hematopoietin cytokine receptor superfamily, functions as a homodimer and requires the recruitment of cytosolic protein tyrosine kinases (PTKs) ... | |||
TMPY-02802 | GNG13 Protein, Human, Recombinant (His) | Human | E. coli |
GNG13 is a subunit of heterotrimeric G proteins which consist of alpha, beta, and gamma subunits. Heterotrimeric G proteins are membrane-bound GTPases that are linked to 7-TM receptors. They function as signal transducer... | |||
TMPY-03280 | RAMP3 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
RAMP3 belongs to the RAMP family. Members of this family are single-transmembrane-domain proteins, called receptor (calcitonin) activity modifying proteins (RAMPs). RAMPs have a wide biological distribution; high concent... | |||
TMPK-00743 | LGR-5 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
G protein-coupled receptor 5 (LGR5), known as a stem cell marker for colon cancer and gastric cancer, can serve as a novel GSC marker involved in EMT and a therapeutic target in glioma.LGR5 is a new functional GSC marker... | |||
TMPY-04555 | GRK5 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
G protein-coupled receptor kinase 5, also known as G protein-coupled receptor kinase GRK5 and GRK5, is a member of the protein kinase superfamily, AGC Ser/Thr protein kinase family, and GPRK subfamily. GRKs specifically ... | |||
TMPY-04409 | GRK6 Protein, Human, Recombinant (His & GST) | Human | Baculovirus Insect Cells |
G protein-coupled receptor kinase 6, also known as G protein-coupled receptor kinase GRK6, GRK6, and GPRK6, is a lipid-anchor protein that belongs to the protein kinase superfamily, AGC Ser/Thr protein kinase family, and... | |||
TMPJ-01202 | LYG2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Lysozyme G-Like Protein 2 (LYG2) is a secreted protein that belongs to the glycosyl hydrolase 23 family. LYG2 contains one SLT domain, one protein domain present in bacterial lytic transglycosylase (SLT) and in eukaryoti... | |||
TMPY-01683 | CD97 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
CD97 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 68.2 kDa and the accession number is P48960-2. | |||
TMPY-02805 | GNGT1 Protein, Human, Recombinant (His) | Human | E. coli |
GNGT1 is a subunit of transducin. Heterotrimeric G proteins consist of alpha, beta, and gamma subunits. They are membrane-bound GTPases that are linked to 7-TM receptors. They function as signal transducers for the 7-tra... | |||
TMPY-01365 | CD97 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
CD97 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 42.6 kDa and the accession number is P48960-2. | |||
TMPJ-01304 | C1QTNF1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
C1QTNF1 is a secreted protein,contains 1 C1q domain and 1 collagen-like domain. C1qTNF proteins constitute a highly conserved family of Acrp30/Adiponectin paralogs that share a modular organization comprising an N-termin... | |||
TMPK-01193 | GPRC5D Protein-VLP, Mouse, Recombinant | Mouse | HEK293 Cells |
Chimeric antigen receptor (CAR) T cells, a type of cell-based immunotherapy, have shown some promising results in multiple myeloma, a bone marrow cancer.The orphan G protein–coupled receptor, class C group 5 member D (GP... | |||
TMPK-00528 | GPRC5D Protein-VLP, Cynomolgus, Recombinant | Cynomolgus | HEK293 Cells |
Chimeric antigen receptor (CAR) T cells, a type of cell-based immunotherapy, have shown some promising results in multiple myeloma, a bone marrow cancer.The orphan G protein–coupled receptor, class C group 5 member D (GP... | |||
TMPH-01082 | CMKLR1 Protein, Human, Recombinant (His) | Human | E. coli |
CMKLR1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 45.1 kDa and the accession number is Q99788. | |||
TMPH-01733 | DDAH2 Protein, Human, Recombinant (GST & His) | Human | E. coli |
Hydrolyzes N(G),N(G)-dimethyl-L-arginine (ADMA) and N(G)-monomethyl-L-arginine (MMA) which act as inhibitors of NOS. Has therefore a role in the regulation of nitric oxide generation. DDAH2 Protein, Human, Recombinant (G... | |||
TMPY-02276 | GPR56 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
ADGRG1 (Adhesion G Protein-Coupled Receptor G1, also known as GPR56) is a Protein Coding gene. GPR56 is a member of an adhesion G protein-coupled receptor family with a very long N-terminal stalk and seven transmembrane ... | |||
TMPY-02924 | RGS1 Protein, Human, Recombinant (His) | Human | E. coli |
RGS1 (regulator of G-protein signaling 1) has been associated with multiple autoimmune disorders including type I diabetes. RGS1 desensitizes the chemokine receptors CCR7 and CXCR4 that are critical to the localization o... | |||
TMPJ-00283 | Carbonic Anhydrase 9 Protein, Human, Recombinant (Avi & His), Biotinylated | Human | HEK293 Cells |
Carbonic anhydrases IX (CA IX), also known as membrane antigen MN or CA9, is a member of the carbonic anhydrase (CA) family and may be involved in cell proliferation and cellular transformation. CAs are zinc metalloenzym... | |||
TMPY-02717 | GPR37 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
GPR37 (cathepsin Z) is an orphan receptor that belongs to the G-protein coupled receptor 1 family. G protein-coupled receptors are a large protein family comprised of transmembrane receptors that sense molecules outside ... | |||
TMPY-06677 | Bla g 4 Protein, cockroaches, Recombinant | cockroaches | P. pastoris (Yeast) |
Bla g 4 Protein, cockroaches, Recombinant is expressed in P. pastoris yeast expression system. The predicted molecular weight is 30 kDa. | |||
TMPH-03749 | CYSLTR1 Protein, Human, Recombinant (His) | Human | E. coli |
Receptor for cysteinyl leukotrienes mediating bronchoconstriction of individuals with and without asthma. Stimulation by LTD4 results in the contraction and proliferation of smooth muscle, edema, eosinophil migration and... | |||
TMPY-00813 | G-CSF Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
G-CSF Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 45.4 kDa and the accession number is P09919-2. | |||
TMPJ-00091 | G-CSF Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Granulocyte colony-stimulating factor (G-CSF) is a growth factor and an essential cytokine which belongs to the IL-6 superfamily. Granulocyte/macrophage colony-stimulating factors are cytokines that act in hematopoiesis ... | |||
TMPH-03265 | CMKLR2 Protein, Rat, Recombinant (His) | Rat | E. coli |
Receptor for chemoattractant adipokine chemerin/RARRES2 suggesting a role for this receptor in the regulation of inflammation and energy homesotasis. Signals mainly via beta-arrestin pathway. Binding of RARRES2 activates... | |||
TMPH-02612 | CXCR3 Protein, Mouse, Recombinant (His & KSI) | Mouse | E. coli |
Receptor for the C-X-C chemokine CXCL9, CXCL10 and CXCL11 and mediates the proliferation, survival and angiogenic activity of mesangial cells through a heterotrimeric G-protein signaling pathway. Probably promotes cell c... | |||
TMPY-04058 | RGS5 Protein, Human, Recombinant (His) | Human | E. coli |
RGS5 is a member of the RGS superfamily and acts as a negative regulator of heterotrimeric G protein-mediated signalling through G protein-coupled receptors (GPCRs). The regulator of G-protein signaling (RGS) proteins ha... | |||
TMPH-01162 | CXCR3 Protein, Human, Recombinant (GST & His) | Human | E. coli |
CXCR3 Protein, Human, Recombinant (GST & His) is expressed in E. coli. | |||
TMPY-06728 | Bla g 7 Protein, German cockroach, Recombinant | German cockroach | E. coli |
Bla g 7 Protein, German cockroach, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 33.8 kDa. | |||
TMPH-00490 | G-CSF Protein, Canine, Recombinant (His & SUMO) | Canine | E. coli |
G-CSF Protein, Canine, Recombinant (His & SUMO) is expressed in E. coli. | |||
TMPY-06729 | Bla g 9 Protein, German cockroach, Recombinant | German cockroach | E. coli |
Bla g 9 Protein, German cockroach, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 40.8 kDa. | |||
TMPY-00814 | CSF3R/G-CSFR Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
CSF3R/G-CSFR Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 93.3 kDa and the accession number is Q99062-1. | |||
TMPH-00458 | Dac g 3 Protein, Dactylis glomerata, Recombinant (His) | Dactylis glomerata | P. pastoris (Yeast) |
Dac g 3 Protein, Dactylis glomerata, Recombinant (His) is expressed in Yeast. | |||
TMPH-00457 | Dac g 4 Protein, Dactylis glomerata, Recombinant (His) | Dactylis glomerata | E. coli |
Dac g 4 Protein, Dactylis glomerata, Recombinant (His) is expressed in E. coli. | |||
TMPY-05189 | Bla g 1 Protein, Blattella germanica, Recombinant (His) | Blattella germanica | E. coli |
Bla g 1 Protein, Blattella germanica, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 46.8 kDa and the accession number is Q9UAM5. | |||
TMPH-00226 | ATPase subunit g Protein, Bovine, Recombinant (His & Myc) | Bovine | E. coli |
ATPase subunit g Protein, Bovine, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 18.7 kDa and the accession number is Q28852. | |||
TMPH-00459 | Dac g 3 Protein, Dactylis glomerata, Recombinant (His & SUMO) | Dactylis glomerata | E. coli |
Dac g 3 Protein, Dactylis glomerata, Recombinant (His & SUMO) is expressed in E. coli. | |||
TMPH-00046 | Aln g I Protein, Alnus glutinosa, Recombinant (Yeast, His) | European alder | P. pastoris (Yeast) |
Aln g I Protein, Alnus glutinosa, Recombinant (Yeast, His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 19.2 kDa and the accession number is P38948. | |||
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L2700 | Adrenergic Receptor-Targeted Compound Library | 193 compounds | |
A unique collection of 193 bioactive compounds specifically targeting adrenergic receptors, effective tool for screening new drugs or new target identification; | |||
L1500 | GPCR Compound Library | 1940 compounds | |
A unique collection of 1940 GPCR-active agents for high throughput screening and high content screening for GPCR drug discovery, and new GPCR target identification and research; | |||
L2800 | Serotonin Receptor-Targeted Compound Library | 268 compounds | |
A unique collection of 268 compounds targeting serotonin receptors for high throughput screening and high content screening; | |||
L1580 | GPCR Compound Library Plus | 338 compounds | |
Well-chosen 338 GPCR targeting compounds with unique structures; | |||
L2610 | Neurotransmitter Receptor Compound Library | 1513 compounds | |
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening; | |||
L7200 | Calcium Channel Compound Library | 140 compounds | |
A unique collection of 140 calcium channel blockers and agonists for high throughput and high content screening; | |||
L2600 | Neuronal Signaling Compound Library | 2540 compounds | |
A unique collection of 2540 compounds targeting CNS signaling for high throughput screening (HTS) and high content screening (HCS) for new drugs; | |||
L3300 | Histamine & Melatonin Receptor-Targeted Compound Library | 153 compounds | |
A unique collection of 153 compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS) for new drugs; | |||
L7600 | Chemokine Inhibitor Library | 59 compounds | |
A unique collection of 59 chemokines or chemokine receptors targeted compounds for high throughput and high content screening; |