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Search Results for " g protein "

Targets

263

Compounds

21

Natural Products

194

Recombinant Proteins

9

Libraries

Cat No. Product Name Synonyms Targets
T67755 Protein kinase G inhibitor-1 PKA
Protein kinase G inhibitor-1 is a potent Protein kinase G inhibitor, IC50= 0.9 uM.
T9940 Protein kinase G inhibitor-2 Others
Protein kinase G inhibitor-2 exhibits antibacterial, antiviral, and antitumor activities.
TP1902L1 G-Protein antagonist peptide acetate Adrenergic Receptor
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide acetate inhibits the activation of Gi or Go by M2 muscarinic cho...
TP1902 G-Protein antagonist peptide
Substance P-related peptide that inhibits binding of G proteins to their receptors. Competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors.
T14898 CCG-63808 GTPase
CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins. CCG-63808 dose-dependently inhibits the TR-FRET signal between RGS4-AF488 and Tb-Gαo with IC50 values of 1.9 μM.
T14897 CCG-63802 GTPase
CCG-63802 is a reversible inhibitor of the regulator of G-protein signaling (RGS) protein and has the greatest potency at RGS4.
TP2254 GTP-Binding Protein Fragment, G alpha Others
Using specific antisera raised against synthetic peptides, we find that three distinct GTP-binding protein alpha subunits remain bound to the plasma membrane even after activation with nonhydrolyzable GTP analog. Trypsin...
T8818 TC-G 1005 GPCR19
TC-G 1005 is a potent and selective GPBA agonist (EC50 :0.72 nM; hTGR5). Selective for TGR5 over FXR (farnesoid X receptor). Increases plasma GLP-1 levels and reduces blood glucose in mice. Orally available.
T7428 SBI-115 GPCR19
SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5
T4083 BAR501 BAR 501 GPCR19
BAR501 is an effective and specific GPBAR1 agonist (EC50: 1 μM).
TQ0252 BAR502 FXR , GPCR19 , Autophagy
BAR502 is a dual GPBAR1 and FXR agonist (IC50s: 0.4 μM and 2 μM).
T20731 Brilliant blue G-250 BBG,Acid blue 90, Coomassie Brilliant Blue G,Brilliant Blue G P2X Receptor
Brilliant blue G-250 (Acid blue 90, Coomassie Brilliant Blue G) is an antagonist of the P2X7 purinergic receptor.
T4352 SB756050 SB-756050,SB 756050 GPCR19
SB756050 is a specific TGR5 agonist.
T2088 APD668 APD 668 GPR , P450 , Potassium Channel
APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119, respectively.
T6434 CCG-50014 CCG 50014 GTPase
CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.
T16378 Ogerin Others , 5-HT Receptor , Adenosine Receptor
Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice. Ogerin displays inverse agonist and antagonist activity (Ki, 220 nM) at A2A receptor and weak an...
T1793 MBX-2982 GPR
MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.
T21874 CID 2745687 GPR
CID 2745687 is a GPR35 antagonist that inhibited the effects at human GPR35 of cromolyn disodium and zaprinast, two agonists that share an overlapping binding site.
T6843 GDC-0623 G-868,GDC0623,RG 7421,MEK inhibitor 1 Apoptosis , MEK
GDC-0623 (RG 7421) is a potent and ATP-uncompetitive MEK1 inhibitor with Ki of 0.13 nM. Phase 1.
T1824 TGR5 Receptor Agonist GPCR19
TGR5 is a potent TGR5(GPCR19) agonist.
T2701 GSK1292263 GPR
GSK1292263 is a GPR119 agonist and has been investigated for the treatment of DIABETES MELLITUS, TYPE 2.
T22996 ML-191 ERK
ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.
T6313 Go 6983 Goe 6983 PKC
Go 6983 is a pan-PKC inhibitor targeting PKCα, PKCβ, PKCγ, PKCδ, and PKCζ, exhibiting IC50 values of 7 nM, 7 nM, 6 nM, 10 nM, and 60 nM, respectively.
T4626 TC-O 9311 free base GPR
TC-O 9311 is a potent GPR139 agonist.
T22408 Proflavine 3,6-Diaminoacridine Antibacterial
Proflavine (3,6-Diaminoacridine) (3,6-Diaminoacridine) is a disinfectant bacteriostatic against many gram-positive bacteria and is a topical antiseptic used mainly in wound dressings.
T7156 NIBR189 EBI2/GPR183
NIBR189 is a potent and selective antagonist of EBI2 (GPR183) receptor (IC50 of 11 and 15 nM for human and mouse EBI2 receptors, respectively)
T8329 AR 231453 GPR
AR 231453 is a selective and orally available GPR119 agonist,can stimulate β-cell replication and improve islet graft function.
T2036 6-OAU GTPL5846 GPR
6-OAU (GTPL5846)(GTPL5846; 6-n-octylaminouracil) is a surrogate agonist of GPR84; activates human GPR84 in the presence of Gqi5 chimera in HEK293 cells with an EC50 of 105 nM in the PI assay.
T8975 PSB-SB-487 Cannabinoid Receptor
PSB-SB-487 is antagonist of GPR55.
T8571 ML-184 CID2440433 Cannabinoid Receptor
ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.
T3119 JNJ-63533054 JNJ 63533054 GPR
JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.
T3176 APD597 JNJ-38431055 GPR
APD597 (JNJ-38431055) is a GPR119 agonist, used in the treatment of type 2 diabetes.
T21623 AS1269574 AS 1269574 GPR , TRP/TRPV Channel
AS1269574 is a potent, orally available GPR119 agonist. AS1269574(AS 1269574) has the potential for the research of type 2 diabetes.
T22103 ML-193 CID 1261822 Cannabinoid Receptor
ML-193 (CID 1261822) is a potent and selective GPR55 antagonist( IC50 : 221 nM). It shows more than 27-fold selectivity for GPR55 over GPR35, CB1 and CB2, and can improve the motor and the sensorimotor deficits of Parkin...
T23204 PSN 375963 PSN 375963 hydrochloride GPR
PSN 375963 (PSN 375963 hydrochloride) hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.
T9317 TAK-041 NBI-1065846 GPR
TAK-041 (NBI-1065846) is a potent and selective GPR139 agonist.
T0438 Proflavine Hemisulfate 3,6-Diaminoacridine hemisulfate,Proflavin hemisulfate Others , Potassium Channel , DNA , Thrombin , Antibacterial , Autophagy
Proflavine Hemisulfate (3,6-Diaminoacridine hemisulfate) is the hemisulfate salt form of proflavine, an acridine-derived fluorescent contrast and disinfectant agent that can potentially be used for cellular imaging and a...
T4494 CLOZAPINE N-OXIDE Dopamine Receptor , 5-HT Receptor , AChR , Drug Metabolite
Clozapine N-oxide is the major metabolite of Clozapine and is blood-brain barrier permeable. Clozapine N-oxide is an agonist of DREADDs and activates the DREADD receptors hM3Dq and hM4Di. Clozapine N-oxide is also a dopa...
T4478 CID 16020046 C390-0219 Cannabinoid Receptor
CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.
T12883 Fezagepras PBI-4050,Setogepram GPR
Fezagepras (Setogepram) is an orally active GPR40 agonist and is an antagonist or inverse agonist of GPR84 with anti-inflammatory, anti-fibrotic, and anti-proliferative actions.
T28073 MLS1547 MLS000051547,MLS 1547,MLS-1547 Dopamine Receptor
MLS1547 (MLS000051547) is a highly efficacious agonist of G protein-biased dopamine D2 receptor with a Ki of 1.2 μM. MLS1547 stimulates D2R G protein-mediated signaling with EC50 of 0.37 μM in a calcium mobilization assa...
T10363 Arazine N-Acetyl-S-farnesyl-L-cysteine Others
Arazine (N-Acetyl-S-farnesyl-L-cysteine) can be a a substrate for isoprenylcysteine methyltransferase by competing with prenylated G protein or its receptors site. Arazine is a cell-permeable modulator of G protein and G...
T36036 CAY10786 GPR52 antagonist-1 GPR
CAY10786 (GPR52 antagonist-1) is an antagonist of G protein-coupled receptor 52 (GPR52, IC50 = 0.63 μM).
T16519L BIM-46187 4HCl PH-064 4HCl Others
BIM-46187 4HCl (PH-064 4HCl) is a heterotrimeric G-protein complex inhibitor.
T13807 OSIP-486823 CP248 Microtubule Associated , PKA
OSIP-486823(CP248) is a novel and potent microtubule disruptor with affinity for both protein kinase G (PKG) and microtubules.
T7281 F-15599 5-HT Receptor
F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).
T50088 N-phenylthiophene-2-carboximidamide Others
N-phenylthiophene-2-carboximidamide is a thiophene derivative that functions as an inhibitor of protein tyrosine kinases (PTKs) and a ligand for G protein-coupled receptors (GPCRs).
T5100 DJ-V-159 DJ-V159 GPR , Androgen Receptor
DJ-V-159 is a GPRC6A agonist, targeting the G protein-coupled receptor family C group 6 member A (GPRC6A).
T7312 AX20017 Others , Antibacterial
AX20017 is a small-molecule protein kinase G (PknG) inhibitor(IC50 : 0.39 μM). It acts by blocking the proliferation of M. tuberculosis.
T5422 CID 1375606 CID-1375606,CID1375606 Others
CID 1375606 is a surrogate agonist of orphan G protein-coupled receptor GPR27. characterized by a high level of conservation among vertebrates and a predominant expression in the central nervous system.

Compounds

Protein kinase G inhibitor-1
T67755
Synonym:
Target: PKA
Protein kinase G inhibitor-2
T9940
Synonym:
Target: Others
G-Protein antagonist peptide acetate
TP1902L1
Synonym:
Target: Adrenergic Receptor
G-Protein antagonist peptide
TP1902
Synonym:
Target:
CCG-63808
T14898
Synonym:
Target: GTPase
CCG-63802
T14897
Synonym:
Target: GTPase
GTP-Binding Protein Fragment, G alpha
TP2254
Synonym:
Target: Others
TC-G 1005
T8818
Synonym:
Target: GPCR19
SBI-115
T7428
Synonym:
Target: GPCR19
BAR501
T4083
Synonym: BAR 501
Target: GPCR19
BAR502
TQ0252
Synonym:
Target: FXR, GPCR19, Autophagy
Brilliant blue G-250
T20731
Synonym: BBG,Acid blue 90, Coomassie Brilliant Blue G,Brilliant Blue G
Target: P2X Receptor
SB756050
T4352
Synonym: SB-756050,SB 756050
Target: GPCR19
APD668
T2088
Synonym: APD 668
Target: GPR, P450, Potassium Channel
CCG-50014
T6434
Synonym: CCG 50014
Target: GTPase
Ogerin
T16378
Synonym:
Target: Others, 5-HT Receptor, Adenosine Receptor
MBX-2982
T1793
Synonym:
Target: GPR
CID 2745687
T21874
Synonym:
Target: GPR
GDC-0623
T6843
Synonym: G-868,GDC0623,RG 7421,MEK inhibitor 1
Target: Apoptosis, MEK
TGR5 Receptor Agonist
T1824
Synonym:
Target: GPCR19
GSK1292263
T2701
Synonym:
Target: GPR
ML-191
T22996
Synonym:
Target: ERK
Go 6983
T6313
Synonym: Goe 6983
Target: PKC
TC-O 9311 free base
T4626
Synonym:
Target: GPR
Proflavine
T22408
Synonym: 3,6-Diaminoacridine
Target: Antibacterial
NIBR189
T7156
Synonym:
Target: EBI2/GPR183
AR 231453
T8329
Synonym:
Target: GPR
6-OAU
T2036
Synonym: GTPL5846
Target: GPR
PSB-SB-487
T8975
Synonym:
Target: Cannabinoid Receptor
ML-184
T8571
Synonym: CID2440433
Target: Cannabinoid Receptor
JNJ-63533054
T3119
Synonym: JNJ 63533054
Target: GPR
APD597
T3176
Synonym: JNJ-38431055
Target: GPR
AS1269574
T21623
Synonym: AS 1269574
Target: GPR, TRP/TRPV Channel
ML-193
T22103
Synonym: CID 1261822
Target: Cannabinoid Receptor
PSN 375963
T23204
Synonym: PSN 375963 hydrochloride
Target: GPR
TAK-041
T9317
Synonym: NBI-1065846
Target: GPR
Proflavine Hemisulfate
T0438
Synonym: 3,6-Diaminoacridine hemisulfate,Proflavin hemisulfate
Target: Others, Potassium Channel, DNA, Thrombin, Antibacterial, Autophagy
CLOZAPINE N-OXIDE
T4494
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, AChR, Drug Metabolite
CID 16020046
T4478
Synonym: C390-0219
Target: Cannabinoid Receptor
Fezagepras
T12883
Synonym: PBI-4050,Setogepram
Target: GPR
MLS1547
T28073
Synonym: MLS000051547,MLS 1547,MLS-1547
Target: Dopamine Receptor
Arazine
T10363
Synonym: N-Acetyl-S-farnesyl-L-cysteine
Target: Others
CAY10786
T36036
Synonym: GPR52 antagonist-1
Target: GPR
BIM-46187 4HCl
T16519L
Synonym: PH-064 4HCl
Target: Others
OSIP-486823
T13807
Synonym: CP248
Target: Microtubule Associated, PKA
F-15599
T7281
Synonym:
Target: 5-HT Receptor
N-phenylthiophene-2-carboximidamide
T50088
Synonym:
Target: Others
DJ-V-159
T5100
Synonym: DJ-V159
Target: GPR, Androgen Receptor
AX20017
T7312
Synonym:
Target: Others, Antibacterial
CID 1375606
T5422
Synonym: CID-1375606,CID1375606
Target: Others
1 2 3 4 5 6
Cat No. Product Name Synonyms Targets
T6512 G-418 disulfate Geneticin,G418 Sulfate,Antibiotic G-418 sulfate,Geneticin sulfate Antibacterial , Antibiotic
G-418 disulfate (Geneticin sulfate) is an aminoglycoside antibiotic, an inhibitor of protein synthesis with eukaryotic selectivity. G-418 disulfate blocks peptide synthesis by inhibiting peptide chain elongation.
T5077 Deoxycholic acid sodium salt Sodium deoxycholate,Sodium Desoxycholate Endogenous Metabolite , GPCR19
Deoxycholic acid sodium salt (Sodium deoxycholate) can activate the G protein-coupled bile acid receptor TGR5 that stimulates brown adipose tissue (BAT) thermogenic activity.
T2965 Deoxycholic acid Cholorebic,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic Endogenous Metabolite , GPCR19
Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate. It is usually conjugated with glycine or taurine. Deoxycholic acid acts as a detergent to solubilize fats for intestinal absorptio...
TN2268 Tetrahydromagnolol Cannabinoid Receptor , GPR , GABA Receptor
Tetrahydromagnolol can activate cannabinoid (CB) receptors.
T0700 Ursodeoxycholic acid UDCA,Ursodiol Potassium Channel , Endogenous Metabolite
Ursodeoxycholic acid (UDCA) can be used to dissolve gallstones and reduce cholesterol absorption.
T2968 Hyodeoxycholic acid NSC 60672,α-Hyodeoxycholic Acid,HDCA FXR , Endogenous Metabolite , GPCR19
Hyodeoxycholic acid (NSC 60672) has been used in trials studying the treatment of Hypercholesterolemia.
T29078 Ursodeoxycholic acid sodium UDCA Na,UDCA sodium,Sodium Ursodeoxycholate,Ursodiol sodium,Ursodeoxycholic Acid (sodium salt),Ursodeoxycholate sodium FXR , Endogenous Metabolite , GPCR19
Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities. Ursodeoxycholic acid sodium acts as signaling molecule, exerting it...
T14046 Anandamide (5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide Cannabinoid Receptor , Endogenous Metabolite
Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but also other targets (e.g., GPR18/GPR55) in the central nervous sy...
T0508 γ-Aminobutyric acid Gamma-aminobutyric acid,4-Aminobutyric acid,GABA,4-Aminobutanoic acid,Piperidic acid GABA Receptor , Endogenous Metabolite
γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.
T4839 Ac-Ala-OH N-Acetylalanine,N-Acetyl-L-alanine Others , Endogenous Metabolite
Ac-Ala-OH (N-Acetyl-L-alanine) is a substrate for Guanine nucleotide-binding protein G(I)/G(S)/G(O) gamma-2 subunit, Myelin basic protein, GTP-binding nuclear protein Ran, Tropomyosin alpha 4 chain, HIV-1 Rev binding pro...
T20003 Acridone Antibacterial , ABC
Acridone could induce cell apoptosis, inhibited ABCG2 (ATP-binding cassette sub-family G member 2) protein, and adjusted hormone level.
T3S1612 Kuwanon G Moracenin B,Kuwanone G Phosphatase , Antibacterial , Bombesin Receptor , AChR , AChE , Glucosidase
1. Kuwanon G (Moracenin B) as dual inhibitors of PTP1B and α-glucosidase enzymes, as well as insulin sensitizers, it may potentially be utilized as an effective treatment for Type II diabetes mellitus. 2. Kuwanon G has a...
T3232 Higenamine hydrochloride Higenamine HCl,Demethylcoclaurine hydrochloride,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride Adrenergic Receptor
Higenamine hydrochloride (norcoclaurine HCl) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein–coupled receptors, and are the most prominent...
T5065 GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD Monosodium-GMP,cGMP sodium salt,Cyclic GMP PKA
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD (cGMP sodium salt) , also known as cGMP, is a cellular regulatory agent and has been described as a second messenger. Its levels increase in response to a variety of hormones, inc...
T3929 Kaurenoic acid Kauren-19-Oic Acid,kaurenoate,kaur-16-en-18-oic acid Others
Kaurenoic acid (kaurenoate) has anti-inflammatory potential in acetic acid-induced colitis, decreases in MDA level. Kaurenoic acid exerts a uterine relaxant effect acting principally through calcium blockade and in part,...
T17273 YM-254890 Others
YM-254890 inhibits platelet aggregation induced by ADP by blocking the P2Y1 signal transduction pathway (IC50: below 0.6 μM). YM-254890 is a selective Gαq/11 protein inhibitor. YM-254890 displays no inhibition of other G...
T73876 Sanggenon G
Sanggenon G, a cell-permeable and potent inhibitor of X-linked inhibitor of apoptosis protein (XIAP), specifically binds to the XIAP BIR3 domain with a binding affinity of 34.26 μM, thereby enhancing caspase activation [...
TN5580 Rediocide A
Rediocide A, an insecticide, can inhibit calcium mobilization in Drosophila G-protein- coupled receptors (GPCR)s other than methuselah, it can induce GPCR desensitization and internalization, and such effects are mediate...
T38331 Commendamide
Commendamide is a natural bacterial product that was discovered in a screen for commensal bacteria effector genes (Cbegs). Cbeg12 is a bacterial effector gene that encodes for its production. Commendamide is structurally...
T21500 Sphingosine-1-phosphate S1P Endogenous Metabolite , S1P Receptor , LPL Receptor
Sphingosine-1-phosphate (S1P) is an agonist for S1P1-5 receptors and a ligand for GPR3, GPR6, GPR12.Sphingosine-1-phosphate is an intracellular second messenger that mobilises Ca2+ as an extracellular ligand for G-protei...
T38069 Aquastatin A
Aquastatin A is a fungal metabolite originally isolated fromF. aquaeductuumthat has diverse biological activities.1It is active againstS. aureus(MIC = 32 μg/ml) and inhibits enoyl-acyl carrier protein reductase (Fabl; IC...

Natural Products

G-418 disulfate
T6512
Synonym: Geneticin,G418 Sulfate,Antibiotic G-418 sulfate,Geneticin sulfate
Target: Antibacterial, Antibiotic
Deoxycholic acid sodium salt
T5077
Synonym: Sodium deoxycholate,Sodium Desoxycholate
Target: Endogenous Metabolite, GPCR19
Deoxycholic acid
T2965
Synonym: Cholorebic,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic
Target: Endogenous Metabolite, GPCR19
Tetrahydromagnolol
TN2268
Synonym:
Target: Cannabinoid Receptor, GPR, GABA Receptor
Ursodeoxycholic acid
T0700
Synonym: UDCA,Ursodiol
Target: Potassium Channel, Endogenous Metabolite
Hyodeoxycholic acid
T2968
Synonym: NSC 60672,α-Hyodeoxycholic Acid,HDCA
Target: FXR, Endogenous Metabolite, GPCR19
Ursodeoxycholic acid sodium
T29078
Synonym: UDCA Na,UDCA sodium,Sodium Ursodeoxycholate,Ursodiol sodium,Ursodeoxycholic Acid (sodium salt),Ursodeoxycholate sodium
Target: FXR, Endogenous Metabolite, GPCR19
Anandamide
T14046
Synonym: (5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide
Target: Cannabinoid Receptor, Endogenous Metabolite
γ-Aminobutyric acid
T0508
Synonym: Gamma-aminobutyric acid,4-Aminobutyric acid,GABA,4-Aminobutanoic acid,Piperidic acid
Target: GABA Receptor, Endogenous Metabolite
Ac-Ala-OH
T4839
Synonym: N-Acetylalanine,N-Acetyl-L-alanine
Target: Others, Endogenous Metabolite
Acridone
T20003
Synonym:
Target: Antibacterial, ABC
kuwanon G
T3S1612
Synonym: Moracenin B,Kuwanone G
Target: Phosphatase, Antibacterial, Bombesin Receptor, AChR, AChE, Glucosidase
Higenamine hydrochloride
T3232
Synonym: Higenamine HCl,Demethylcoclaurine hydrochloride,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride
Target: Adrenergic Receptor
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD
T5065
Synonym: Monosodium-GMP,cGMP sodium salt,Cyclic GMP
Target: PKA
Kaurenoic acid
T3929
Synonym: Kauren-19-Oic Acid,kaurenoate,kaur-16-en-18-oic acid
Target: Others
YM-254890
T17273
Synonym:
Target: Others
Sanggenon G
T73876
Synonym:
Target:
Rediocide A
TN5580
Synonym:
Target:
Commendamide
T38331
Synonym:
Target:
Sphingosine-1-phosphate
T21500
Synonym: S1P
Target: Endogenous Metabolite, S1P Receptor, LPL Receptor
Aquastatin A
T38069
Synonym:
Target:

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-01885 Human RSV (B1) glycoprotein G/RSV-G Protein (His) RSV HEK293 Cells
Human RSV (B1) glycoprotein G/RSV-G Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27 kDa and the accession number is O36633-1.
TMPY-01082 Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (95% Homology) (His) RSV HEK293 Cells
Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (95% Homology) (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.7 kDa and the accession num...
TMPY-02283 Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (93% Homology) (His) RSV Baculovirus Insect Cells
Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (93% Homology) (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 26.3 kDa and the accession n...
TMPY-00105 Recombinant Protein G E. coli
Protein G is a bacterial cell wall protein expressed at the cell surface of certain group C and group G Streptococcal strains. It has affinity for both Fab- and Fc-fragments of human IgG by independent and separate bindi...
TMPY-06469 Human respiratory syncytial virus (RSV) (B, strain 18537) glycoprotein G Protein (His) RSV HEK293 Cells
Human respiratory syncytial virus (RSV) (B, strain 18537) glycoprotein G Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.40 kDa and the accession number is P20896.
TMPY-06474 Human respiratory syncytial virus (RSV) (strain A2) glycoprotein G Protein (His) RSV HEK293 Cells
Human respiratory syncytial virus (RSV) (strain A2) glycoprotein G Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.97 kDa and the accession number is P03423.
TMPY-05686 Human respiratory syncytial virus (RSV) glycoprotein G Protein (aa 64-321, His) RSV HEK293 Cells
Human respiratory syncytial virus (RSV) glycoprotein G Protein (aa 64-321, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 29.59 kDa and the accession number is A0A076FRQ0.
TMPY-06111 Human respiratory syncytial virus (RSV) (subtype A, strain Long) glycoprotein G Protein (His) RSV HEK293 Cells
Human respiratory syncytial virus (RSV) (subtype A, strain Long) glycoprotein G Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27 kDa and the accession number is P208...
TMPY-05636 G-CSF Protein, Mouse, Recombinant Mouse HEK293 Cells
G-CSF Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 19 kDa and the accession number is P09920.
TMPY-04829 G-CSF Protein, Human, Recombinant Human HEK293 Cells
G-CSF Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 18.7 kDa and the accession number is P09919-2.
TMPY-02312 CSF3R/G-CSFR Protein, Human, Recombinant (His) Human HEK293 Cells
CSF3R/G-CSFR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 68 kDa and the accession number is Q99062-1.
TMPY-00300 Hendra virus (HeV) (isolate Horse/Autralia/Hendra/1994) Glycoprotein Protein (hFc) HEV HEK293 Cells
Hendra virus (HeV) (isolate Horse/Autralia/Hendra/1994) Glycoprotein Protein (hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 86.3 kDa and the accession number is O89343.
TMPH-00510 DT3C Protein, Recombinant (His) Corynephage beta E. coli
DT3C Protein, Recombinant (His) is expressed in E. coli.
TMPK-00876 G-CSFR/CD114 Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
The Granulocyte Colony-Stimulating Factor (G-CSF) receptor, a member of the hematopoietin cytokine receptor superfamily, functions as a homodimer and requires the recruitment of cytosolic protein tyrosine kinases (PTKs) ...
TMPY-02802 GNG13 Protein, Human, Recombinant (His) Human E. coli
GNG13 is a subunit of heterotrimeric G proteins which consist of alpha, beta, and gamma subunits. Heterotrimeric G proteins are membrane-bound GTPases that are linked to 7-TM receptors. They function as signal transducer...
TMPY-03280 RAMP3 Protein, Human, Recombinant (hFc) Human HEK293 Cells
RAMP3 belongs to the RAMP family. Members of this family are single-transmembrane-domain proteins, called receptor (calcitonin) activity modifying proteins (RAMPs). RAMPs have a wide biological distribution; high concent...
TMPK-00743 LGR-5 Protein, Human, Recombinant (hFc) Human HEK293 Cells
G protein-coupled receptor 5 (LGR5), known as a stem cell marker for colon cancer and gastric cancer, can serve as a novel GSC marker involved in EMT and a therapeutic target in glioma.LGR5 is a new functional GSC marker...
TMPY-04555 GRK5 Protein, Human, Recombinant (His) Human Baculovirus Insect Cells
G protein-coupled receptor kinase 5, also known as G protein-coupled receptor kinase GRK5 and GRK5, is a member of the protein kinase superfamily, AGC Ser/Thr protein kinase family, and GPRK subfamily. GRKs specifically ...
TMPY-04409 GRK6 Protein, Human, Recombinant (His & GST) Human Baculovirus Insect Cells
G protein-coupled receptor kinase 6, also known as G protein-coupled receptor kinase GRK6, GRK6, and GPRK6, is a lipid-anchor protein that belongs to the protein kinase superfamily, AGC Ser/Thr protein kinase family, and...
TMPJ-01202 LYG2 Protein, Human, Recombinant (His) Human HEK293 Cells
Lysozyme G-Like Protein 2 (LYG2) is a secreted protein that belongs to the glycosyl hydrolase 23 family. LYG2 contains one SLT domain, one protein domain present in bacterial lytic transglycosylase (SLT) and in eukaryoti...
TMPY-01683 CD97 Protein, Human, Recombinant (hFc) Human HEK293 Cells
CD97 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 68.2 kDa and the accession number is P48960-2.
TMPY-02805 GNGT1 Protein, Human, Recombinant (His) Human E. coli
GNGT1 is a subunit of transducin. Heterotrimeric G proteins consist of alpha, beta, and gamma subunits. They are membrane-bound GTPases that are linked to 7-TM receptors. They function as signal transducers for the 7-tra...
TMPY-01365 CD97 Protein, Human, Recombinant (His) Human HEK293 Cells
CD97 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 42.6 kDa and the accession number is P48960-2.
TMPJ-01304 C1QTNF1 Protein, Human, Recombinant (His) Human HEK293 Cells
C1QTNF1 is a secreted protein,contains 1 C1q domain and 1 collagen-like domain. C1qTNF proteins constitute a highly conserved family of Acrp30/Adiponectin paralogs that share a modular organization comprising an N-termin...
TMPK-01193 GPRC5D Protein-VLP, Mouse, Recombinant Mouse HEK293 Cells
Chimeric antigen receptor (CAR) T cells, a type of cell-based immunotherapy, have shown some promising results in multiple myeloma, a bone marrow cancer.The orphan G protein–coupled receptor, class C group 5 member D (GP...
TMPK-00528 GPRC5D Protein-VLP, Cynomolgus, Recombinant Cynomolgus HEK293 Cells
Chimeric antigen receptor (CAR) T cells, a type of cell-based immunotherapy, have shown some promising results in multiple myeloma, a bone marrow cancer.The orphan G protein–coupled receptor, class C group 5 member D (GP...
TMPH-01082 CMKLR1 Protein, Human, Recombinant (His) Human E. coli
CMKLR1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 45.1 kDa and the accession number is Q99788.
TMPH-01733 DDAH2 Protein, Human, Recombinant (GST & His) Human E. coli
Hydrolyzes N(G),N(G)-dimethyl-L-arginine (ADMA) and N(G)-monomethyl-L-arginine (MMA) which act as inhibitors of NOS. Has therefore a role in the regulation of nitric oxide generation. DDAH2 Protein, Human, Recombinant (G...
TMPY-02276 GPR56 Protein, Human, Recombinant (His) Human HEK293 Cells
ADGRG1 (Adhesion G Protein-Coupled Receptor G1, also known as GPR56) is a Protein Coding gene. GPR56 is a member of an adhesion G protein-coupled receptor family with a very long N-terminal stalk and seven transmembrane ...
TMPY-02924 RGS1 Protein, Human, Recombinant (His) Human E. coli
RGS1 (regulator of G-protein signaling 1) has been associated with multiple autoimmune disorders including type I diabetes. RGS1 desensitizes the chemokine receptors CCR7 and CXCR4 that are critical to the localization o...
TMPJ-00283 Carbonic Anhydrase 9 Protein, Human, Recombinant (Avi & His), Biotinylated Human HEK293 Cells
Carbonic anhydrases IX (CA IX), also known as membrane antigen MN or CA9, is a member of the carbonic anhydrase (CA) family and may be involved in cell proliferation and cellular transformation. CAs are zinc metalloenzym...
TMPY-02717 GPR37 Protein, Human, Recombinant (His) Human HEK293 Cells
GPR37 (cathepsin Z) is an orphan receptor that belongs to the G-protein coupled receptor 1 family. G protein-coupled receptors are a large protein family comprised of transmembrane receptors that sense molecules outside ...
TMPY-06677 Bla g 4 Protein, cockroaches, Recombinant cockroaches P. pastoris (Yeast)
Bla g 4 Protein, cockroaches, Recombinant is expressed in P. pastoris yeast expression system. The predicted molecular weight is 30 kDa.
TMPH-03749 CYSLTR1 Protein, Human, Recombinant (His) Human E. coli
Receptor for cysteinyl leukotrienes mediating bronchoconstriction of individuals with and without asthma. Stimulation by LTD4 results in the contraction and proliferation of smooth muscle, edema, eosinophil migration and...
TMPY-00813 G-CSF Protein, Human, Recombinant (hFc) Human HEK293 Cells
G-CSF Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 45.4 kDa and the accession number is P09919-2.
TMPJ-00091 G-CSF Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Granulocyte colony-stimulating factor (G-CSF) is a growth factor and an essential cytokine which belongs to the IL-6 superfamily. Granulocyte/macrophage colony-stimulating factors are cytokines that act in hematopoiesis ...
TMPH-03265 CMKLR2 Protein, Rat, Recombinant (His) Rat E. coli
Receptor for chemoattractant adipokine chemerin/RARRES2 suggesting a role for this receptor in the regulation of inflammation and energy homesotasis. Signals mainly via beta-arrestin pathway. Binding of RARRES2 activates...
TMPH-02612 CXCR3 Protein, Mouse, Recombinant (His & KSI) Mouse E. coli
Receptor for the C-X-C chemokine CXCL9, CXCL10 and CXCL11 and mediates the proliferation, survival and angiogenic activity of mesangial cells through a heterotrimeric G-protein signaling pathway. Probably promotes cell c...
TMPY-04058 RGS5 Protein, Human, Recombinant (His) Human E. coli
RGS5 is a member of the RGS superfamily and acts as a negative regulator of heterotrimeric G protein-mediated signalling through G protein-coupled receptors (GPCRs). The regulator of G-protein signaling (RGS) proteins ha...
TMPH-01162 CXCR3 Protein, Human, Recombinant (GST & His) Human E. coli
CXCR3 Protein, Human, Recombinant (GST & His) is expressed in E. coli.
TMPY-06728 Bla g 7 Protein, German cockroach, Recombinant German cockroach E. coli
Bla g 7 Protein, German cockroach, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 33.8 kDa.
TMPH-00490 G-CSF Protein, Canine, Recombinant (His & SUMO) Canine E. coli
G-CSF Protein, Canine, Recombinant (His & SUMO) is expressed in E. coli.
TMPY-06729 Bla g 9 Protein, German cockroach, Recombinant German cockroach E. coli
Bla g 9 Protein, German cockroach, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 40.8 kDa.
TMPY-00814 CSF3R/G-CSFR Protein, Human, Recombinant (hFc) Human HEK293 Cells
CSF3R/G-CSFR Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 93.3 kDa and the accession number is Q99062-1.
TMPH-00458 Dac g 3 Protein, Dactylis glomerata, Recombinant (His) Dactylis glomerata P. pastoris (Yeast)
Dac g 3 Protein, Dactylis glomerata, Recombinant (His) is expressed in Yeast.
TMPH-00457 Dac g 4 Protein, Dactylis glomerata, Recombinant (His) Dactylis glomerata E. coli
Dac g 4 Protein, Dactylis glomerata, Recombinant (His) is expressed in E. coli.
TMPY-05189 Bla g 1 Protein, Blattella germanica, Recombinant (His) Blattella germanica E. coli
Bla g 1 Protein, Blattella germanica, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 46.8 kDa and the accession number is Q9UAM5.
TMPH-00226 ATPase subunit g Protein, Bovine, Recombinant (His & Myc) Bovine E. coli
ATPase subunit g Protein, Bovine, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 18.7 kDa and the accession number is Q28852.
TMPH-00459 Dac g 3 Protein, Dactylis glomerata, Recombinant (His & SUMO) Dactylis glomerata E. coli
Dac g 3 Protein, Dactylis glomerata, Recombinant (His & SUMO) is expressed in E. coli.
TMPH-00046 Aln g I Protein, Alnus glutinosa, Recombinant (Yeast, His) European alder P. pastoris (Yeast)
Aln g I Protein, Alnus glutinosa, Recombinant (Yeast, His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 19.2 kDa and the accession number is P38948.
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Human RSV (B1) glycoprotein G/RSV-G Protein (His)
TMPY-01885
Species: RSV
Expression System: HEK293 Cells
Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (95% Homology) (His)
TMPY-01082
Species: RSV
Expression System: HEK293 Cells
Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (93% Homology) (His)
TMPY-02283
Species: RSV
Expression System: Baculovirus Insect Cells
Recombinant Protein G
TMPY-00105
Species:
Expression System: E. coli
Human respiratory syncytial virus (RSV) (B, strain 18537) glycoprotein G Protein (His)
TMPY-06469
Species: RSV
Expression System: HEK293 Cells
Human respiratory syncytial virus (RSV) (strain A2) glycoprotein G Protein (His)
TMPY-06474
Species: RSV
Expression System: HEK293 Cells
Human respiratory syncytial virus (RSV) glycoprotein G Protein (aa 64-321, His)
TMPY-05686
Species: RSV
Expression System: HEK293 Cells
Human respiratory syncytial virus (RSV) (subtype A, strain Long) glycoprotein G Protein (His)
TMPY-06111
Species: RSV
Expression System: HEK293 Cells
G-CSF Protein, Mouse, Recombinant
TMPY-05636
Species: Mouse
Expression System: HEK293 Cells
G-CSF Protein, Human, Recombinant
TMPY-04829
Species: Human
Expression System: HEK293 Cells
CSF3R/G-CSFR Protein, Human, Recombinant (His)
TMPY-02312
Species: Human
Expression System: HEK293 Cells
Hendra virus (HeV) (isolate Horse/Autralia/Hendra/1994) Glycoprotein Protein (hFc)
TMPY-00300
Species: HEV
Expression System: HEK293 Cells
DT3C Protein, Recombinant (His)
TMPH-00510
Species: Corynephage beta
Expression System: E. coli
G-CSFR/CD114 Protein, Mouse, Recombinant (His)
TMPK-00876
Species: Mouse
Expression System: HEK293 Cells
GNG13 Protein, Human, Recombinant (His)
TMPY-02802
Species: Human
Expression System: E. coli
RAMP3 Protein, Human, Recombinant (hFc)
TMPY-03280
Species: Human
Expression System: HEK293 Cells
LGR-5 Protein, Human, Recombinant (hFc)
TMPK-00743
Species: Human
Expression System: HEK293 Cells
GRK5 Protein, Human, Recombinant (His)
TMPY-04555
Species: Human
Expression System: Baculovirus Insect Cells
GRK6 Protein, Human, Recombinant (His & GST)
TMPY-04409
Species: Human
Expression System: Baculovirus Insect Cells
LYG2 Protein, Human, Recombinant (His)
TMPJ-01202
Species: Human
Expression System: HEK293 Cells
CD97 Protein, Human, Recombinant (hFc)
TMPY-01683
Species: Human
Expression System: HEK293 Cells
GNGT1 Protein, Human, Recombinant (His)
TMPY-02805
Species: Human
Expression System: E. coli
CD97 Protein, Human, Recombinant (His)
TMPY-01365
Species: Human
Expression System: HEK293 Cells
C1QTNF1 Protein, Human, Recombinant (His)
TMPJ-01304
Species: Human
Expression System: HEK293 Cells
GPRC5D Protein-VLP, Mouse, Recombinant
TMPK-01193
Species: Mouse
Expression System: HEK293 Cells
GPRC5D Protein-VLP, Cynomolgus, Recombinant
TMPK-00528
Species: Cynomolgus
Expression System: HEK293 Cells
CMKLR1 Protein, Human, Recombinant (His)
TMPH-01082
Species: Human
Expression System: E. coli
DDAH2 Protein, Human, Recombinant (GST & His)
TMPH-01733
Species: Human
Expression System: E. coli
GPR56 Protein, Human, Recombinant (His)
TMPY-02276
Species: Human
Expression System: HEK293 Cells
RGS1 Protein, Human, Recombinant (His)
TMPY-02924
Species: Human
Expression System: E. coli
Carbonic Anhydrase 9 Protein, Human, Recombinant (Avi & His), Biotinylated
TMPJ-00283
Species: Human
Expression System: HEK293 Cells
GPR37 Protein, Human, Recombinant (His)
TMPY-02717
Species: Human
Expression System: HEK293 Cells
Bla g 4 Protein, cockroaches, Recombinant
TMPY-06677
Species: cockroaches
Expression System: P. pastoris (Yeast)
CYSLTR1 Protein, Human, Recombinant (His)
TMPH-03749
Species: Human
Expression System: E. coli
G-CSF Protein, Human, Recombinant (hFc)
TMPY-00813
Species: Human
Expression System: HEK293 Cells
G-CSF Protein, Mouse, Recombinant (His)
TMPJ-00091
Species: Mouse
Expression System: HEK293 Cells
CMKLR2 Protein, Rat, Recombinant (His)
TMPH-03265
Species: Rat
Expression System: E. coli
CXCR3 Protein, Mouse, Recombinant (His & KSI)
TMPH-02612
Species: Mouse
Expression System: E. coli
RGS5 Protein, Human, Recombinant (His)
TMPY-04058
Species: Human
Expression System: E. coli
CXCR3 Protein, Human, Recombinant (GST & His)
TMPH-01162
Species: Human
Expression System: E. coli
Bla g 7 Protein, German cockroach, Recombinant
TMPY-06728
Species: German cockroach
Expression System: E. coli
G-CSF Protein, Canine, Recombinant (His & SUMO)
TMPH-00490
Species: Canine
Expression System: E. coli
Bla g 9 Protein, German cockroach, Recombinant
TMPY-06729
Species: German cockroach
Expression System: E. coli
CSF3R/G-CSFR Protein, Human, Recombinant (hFc)
TMPY-00814
Species: Human
Expression System: HEK293 Cells
Dac g 3 Protein, Dactylis glomerata, Recombinant (His)
TMPH-00458
Species: Dactylis glomerata
Expression System: P. pastoris (Yeast)
Dac g 4 Protein, Dactylis glomerata, Recombinant (His)
TMPH-00457
Species: Dactylis glomerata
Expression System: E. coli
Bla g 1 Protein, Blattella germanica, Recombinant (His)
TMPY-05189
Species: Blattella germanica
Expression System: E. coli
ATPase subunit g Protein, Bovine, Recombinant (His & Myc)
TMPH-00226
Species: Bovine
Expression System: E. coli
Dac g 3 Protein, Dactylis glomerata, Recombinant (His & SUMO)
TMPH-00459
Species: Dactylis glomerata
Expression System: E. coli
Aln g I Protein, Alnus glutinosa, Recombinant (Yeast, His)
TMPH-00046
Species: European alder
Expression System: P. pastoris (Yeast)
Cat No. Product Name
L2700 Adrenergic Receptor-Targeted Compound Library

193 compounds
A unique collection of 193 bioactive compounds specifically targeting adrenergic receptors, effective tool for screening new drugs or new target identification;
L1500 GPCR Compound Library

1940 compounds
A unique collection of 1940 GPCR-active agents for high throughput screening and high content screening for GPCR drug discovery, and new GPCR target identification and research;
L2800 Serotonin Receptor-Targeted Compound Library

268 compounds
A unique collection of 268 compounds targeting serotonin receptors for high throughput screening and high content screening;
L1580 GPCR Compound Library Plus

338 compounds
Well-chosen 338 GPCR targeting compounds with unique structures;
L2610 Neurotransmitter Receptor Compound Library

1513 compounds
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening
L7200 Calcium Channel Compound Library

140 compounds
A unique collection of 140 calcium channel blockers and agonists for high throughput and high content screening;
L2600 Neuronal Signaling Compound Library

2540 compounds
A unique collection of 2540 compounds targeting CNS signaling for high throughput screening (HTS) and high content screening (HCS) for new drugs;
L3300 Histamine & Melatonin Receptor-Targeted Compound Library

153 compounds
A unique collection of 153 compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS) for new drugs;
L7600 Chemokine Inhibitor Library

59 compounds
A unique collection of 59 chemokines or chemokine receptors targeted compounds for high throughput and high content screening;
TargetMol